NANOSIZED ANTIBODY PIPELINE

NanoAbs: Significant Advantages

Alpaca-derived nanosized antibodies (NanoAbs), also known as VHH-antibodies*, exhibit potential as biobetter therapies for a wide range of diseases. Scinai is developing NanoAbs addressing diseases with large unmet medical needs and attractive commercial opportunities, such as psoriasis and asthma.

Human mAb cartoon

Human monoclonal antibody (mAb)

Alpaca-derived VHH Ab

Alpaca-derived NanoAb

Platform Value Proposition

NanoAbs’ unique physicochemical attributes can generate multiple crucial advantages vs human monoclonal antibodies (mAbs)

Manufacturing

  • X10 active pharmaceutical ingredient (API) per gram of manufactured protein vs. mAbs

  • Faster and lower cost production in yeast (pichia) vs mammalian cells

R&D

  • Quicker antibody discovery and optimization due to massive libraries

  • De-risked pipeline development leveraging approved mAb targets

Product

  • Hyper-thermostable = longer shelf life, easier storage & distribution

  • Superior specificity & affinity to target potentially enables lower dose, fewer adverse events, lower cost

  • Adaptable half life

Patient Safety & Convenience

  • Multiple, easier routes of administration

  • Lower immunogenicity

  • Fewer contraindications

  • Potentially safer & lower dose

Leading Scientific Collaborators

From the world-renowned Max Planck Institute for Multidisciplinary Sciences and University Medical Center Göttingen, Germany

Professor Dr. Dirk Görlich

Professor & Director at Max Planck Institute for Multidisciplinary Sciences

2024 Louis-Jeantet Prize & 2022 WLA Prize

Professor Dr. Matthias Dobbelstein

Max Planck Institute Fellow, Professor and Department Head at the University of Göttingen

Scinai’s scientific partners are leaders in designing and optimizing NanoAbs.

The NanoAbs exhibit strong neutralization at picomolar levels of concentration; Hyperthermostability to 95°C (200°F); and potential for convenient administration via inhalation and intradermal injection.

Through the Max Planck alpaca farm in Göttingen, our partners quickly generate massive antibody libraries, and then select optimum candidates in the lab leveraging unique know-how.

Neutralization of SARS-CoV-2 by highly potent, hyper-thermostable, & mutation-tolerant nanobodies | EMBO Journal

Authored by our scientific partners at the Max Planck Institute for Multidisciplinary Sciences and University Medical Center Göttingen, Germany.

Our NanoAb exhibit a strong competitive edge over existing therapies. For example, the anti-Sars-COV-2 NanoAbs exhibit superior affinity to the target, neutralizing the virus, in-vitro, at drug concentrations about 100-times lower than those required by currently commercially available monoclonal antibodies. This may lead to increased efficacy, reduced side effects, and allow production at a lower cost. In addition, the NanoAbs’ small size and hyper-thermostability at 95°C (200°F) potentially enables administration through inhalation and longer shelf life, and potentially avoids the need for enhanced cold chain storage and transport. Together, these attributes are designed to create significant competitive advantages.

https://doi.org/10.15252/embj.2021107985

NanoAbs feature a favorable path to market compared to risks associated with traditional drug development:

  • Molecular Target: Validated by existing but sub-optimal antibody therapies

  • Mechanism of Action: Well understood

  • Commercial: Strong demand for available antibody therapies, and underserved populations

  • Validated Clinical Use: The first commercial VHH-antibody is blood disorder therapy Caplacizuma, developed by Ablynx, a company acquired by Sanofi in 2018 for $4.8B

Derisked Drug Development